Recording Webinar

Recording Webinar The Dynamics of Compound Profiling: Using Signaling Kinetic Assays to Shape Early-Stage Drug Discovery

06/05/2021

The Dynamics of Compound Profiling: Using Signaling Kinetic Assays to Shape Early-Stage Drug DiscoveryIn vitro early-stage compound profiling often focuses on single timepoint measurements of drug action. However, in vivo, drug action occurs not at equilibrium, but within a highly dynamic system. This webinar will explore how measuring the kinetics of drug-target interaction and signaling can help optimize functional compound properties, using NanoBRET™ and NanoBiT® technologies. The webinar will include a panel Q&A session after their presentations.

You will learn about:

  • Realtime measurements of binding and signaling kinetics
  • Mapping therapeutic efforts to patterns of downstream cellular signaling over time
  • Studying signaling kinetics at an early stage to inform lead optimization

Registration link : https://bit.ly/3xNg25e

                             Free Registration

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